GSK046 [Cas No. 2474876-09-8]
Catalog No：TA-T8932
Manufacturer：TargetMol
Synonyms：iBET-BD2
CAS No.：2474876-09-8
Formula：C23H27FN2O4
MWt：414.48
€187,00 – €2.124,00
| Name: | GSK046 |
| Category: | Biochemicals |
| Description: | GSK046 is a potent, selective and orally active BD2 bromodomain inhibitor of the BET proteins(IC50s of 264 nM (BRD2 BD2), 98 nM (BRD3 BD2), 49 nM (BRD4 BD2) and 214 nM (BRDT BD2), respectively). It has immunomodulatory activity. |
| Pathway: | Chromatin/Epigenetic |
| Target: | Epigenetic Reader Domain |
| Receptor: | BRD2-BD2,BRD3-BD2,BRD4-BD2,BRDT-BD2 |
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